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Drug Resistance Resulting from Kinase Dimerization Is Rationalized by Thermodynamic Factors Describing Allosteric Inhibitor Effects
Kholodenko, Boris N.
Kholodenko, Boris N.
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Keywords
Allosteric inhibitor effects
Allosteric kinase activation
drug-facilitated dimerization
BRAF
CRAF
drug resistance
Kinase dimerization
Allosteric inhibitor effects
Allosteric kinase activation
drug-facilitated dimerization
BRAF
CRAF
drug resistance
Kinase dimerization
Allosteric inhibitor effects